SCHEMBL8628065

SCHEMBL8628065

COc1ccc(S(=O)(=O)Nc2cccc(C)c2NC(=O)c2ccc(F)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 2/20 0.58
KEAP1 Q14145 1/20 0.56
STAT3 P40763 1/20 0.55
TSHR P16473 2/20 0.54
HDAC3 O15379 4/20 0.54
NCOR2 Q9Y618 4/20 0.54
HDAC2 Q92769 3/20 0.54
ALDH1A1 P00352 4/20 0.53
KDM4E B2RXH2 3/20 0.53
TUBB4A P04350 1/20 0.52
TUBB P07437 1/20 0.52
TUBA3C P0DPH7 1/20 0.52
TUBA1B P68363 1/20 0.52
TUBA4A P68366 1/20 0.52
TUBB4B P68371 1/20 0.52
TUBB3 Q13509 1/20 0.52
TUBB2A Q13885 1/20 0.52
TUBB8 Q3ZCM7 1/20 0.52
TUBA3E Q6PEY2 1/20 0.52
TUBA1A Q71U36 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8666558 0.87 SMN1; SMN2 (0.61) FFAR4KEAP1TSHRHDAC3NCOR2
SCHEMBL8627623 0.85 F10 (0.64) KEAP1STAT3HDAC3NCOR2HDAC2
SCHEMBL8622517 0.82 FFAR4 (0.55) FFAR4KEAP1TSHRALDH1A1KDM4E
SCHEMBL7249253 0.80 F10 (0.69) HDAC3HDAC2ALDH1A1KMT2AMAPT
SCHEMBL8625140 0.80 MAPT (0.59) FFAR4KEAP1ALDH1A1LMNAMAPT
SCHEMBL27181622 0.78 KMT2A (0.75) STAT3ALDH1A1KDM4ELMNAKMT2A
SCHEMBL27180643 0.78 KMT2A (0.75) STAT3ALDH1A1KDM4ELMNAKMT2A
SCHEMBL6935548 0.77 ALDH1A1 (0.65) HDAC3HDAC2ALDH1A1KDM4ECYP2C9
SCHEMBL27180903 0.77 LMNA (0.62) FFAR4STAT3HDAC3NCOR2HDAC2
SCHEMBL8626446 0.77 STAT3 (0.63) KEAP1STAT3HDAC3NCOR2HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610320-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-03-11 US claimed
EP-0472053-B1 Sulfonamide derivatives EISAI CO LTD (JP) 1998-06-17 EP disclosed
US-5610304-A Pyrimidinyl or pyridinyl sulfonamide substituted compounds EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5610320-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5434172-A Antitumor EISAI CO., LTD. (JP) 1995-07-18 US disclosed
US-5332751-A Antitumor EISAI CO., LTD. (JP) 1994-07-26 US disclosed
US-5292758-A Sulfonamide derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
US-5250549-A Antitumor agents EISAI CO., LTD. (JP) 1993-10-05 US disclosed
EP-0472053-A2 Sulfonamide derivatives Eisai Co., Ltd. (JP) 1992-02-26 EP disclosed