SCHEMBL8666558

SCHEMBL8666558

COc1ccc(S(=O)(=O)Nc2cccc(C)c2NC(=O)c2ccncc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.61
L3MBTL1 Q9Y468 2/20 0.60
FFAR4 Q5NUL3 1/20 0.58
KEAP1 Q14145 1/20 0.56
CCR9 P51686 1/20 0.53
TUBB4A P04350 1/20 0.52
TUBB P07437 1/20 0.52
TUBA3C P0DPH7 1/20 0.52
TUBA1B P68363 1/20 0.52
TUBA4A P68366 1/20 0.52
TUBB4B P68371 1/20 0.52
TUBB3 Q13509 1/20 0.52
TUBB2A Q13885 1/20 0.52
TUBB8 Q3ZCM7 1/20 0.52
TUBA3E Q6PEY2 1/20 0.52
TUBA1A Q71U36 1/20 0.52
TUBA1C Q9BQE3 1/20 0.52
TUBB6 Q9BUF5 1/20 0.52
TUBB2B Q9BVA1 1/20 0.52
TUBB1 Q9H4B7 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8622517 0.89 FFAR4 (0.55) SMN1; SMN2FFAR4KEAP1LMNAPKM
SCHEMBL8628065 0.87 FFAR4 (0.58) FFAR4KEAP1TUBB4ATUBBTUBA3C
SCHEMBL8626468 0.85 SMN1; SMN2 (0.69) SMN1; SMN2L3MBTL1KEAP1CCR9TUBB4A
SCHEMBL8625140 0.84 MAPT (0.59) SMN1; SMN2L3MBTL1FFAR4KEAP1CCR9
SCHEMBL7249253 0.78 F10 (0.69) SMN1; SMN2PKMALDH1A1MEN1KMT2A
SCHEMBL8625192 0.76 F10 (0.67) SMN1; SMN2L3MBTL1KEAP1TUBB4ATUBB
SCHEMBL6359170 0.75 MEN1 (0.68) SMN1; SMN2L3MBTL1CCR9LMNAPKM
SCHEMBL6935548 0.75 ALDH1A1 (0.65) SMN1; SMN2PKMALDH1A1MEN1KMT2A
SCHEMBL8626192 0.74 KEAP1 (0.56) SMN1; SMN2L3MBTL1KEAP1CCR9TUBB4A
SCHEMBL8623537 0.74 KEAP1 (0.56) SMN1; SMN2L3MBTL1KEAP1CCR9TUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0472053-B1 Sulfonamide derivatives EISAI CO LTD (JP) 1998-06-17 EP disclosed
US-5610304-A Pyrimidinyl or pyridinyl sulfonamide substituted compounds EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5610320-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5434172-A Antitumor EISAI CO., LTD. (JP) 1995-07-18 US disclosed
US-5332751-A Antitumor EISAI CO., LTD. (JP) 1994-07-26 US disclosed
US-5292758-A Sulfonamide derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
US-5250549-A Antitumor agents EISAI CO., LTD. (JP) 1993-10-05 US disclosed
EP-0472053-A2 Sulfonamide derivatives Eisai Co., Ltd. (JP) 1992-02-26 EP disclosed