SCHEMBL8628090

SCHEMBL8628090

COC(=O)C#CC(=O)c1cccc(OC)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.59
CES1 P23141 1/20 0.59
PARP1 P09874 1/20 0.56
NPC1 O15118 7/20 0.54
RAB9A P51151 7/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
SMN1; SMN2 Q16637 5/20 0.51
TSHR P16473 3/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TAS1R3 Q7RTX0 1/20 0.50
TAS1R1 Q7RTX1 1/20 0.50
POLB P06746 1/20 0.49
BLM P54132 1/20 0.49
TP53 P04637 3/20 0.49
ALDH1A1 P00352 2/20 0.49
KCNK3 O14649 1/20 0.49
KCNK9 Q9NPC2 1/20 0.49
KDM4E B2RXH2 1/20 0.49
NFKB1 P19838 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24081297 0.83 CES2 (0.62) CES2CES1PARP1NPC1RAB9A
SCHEMBL8626440 0.82 HDAC8 (0.50) PARP1NPC1RAB9AMEN1KMT2A
SCHEMBL8630144 0.81 ERCC5 (0.47) PARP1NPC1RAB9AMEN1KMT2A
SCHEMBL8626139 0.80 APP (0.55) CES2CES1PARP1NPC1RAB9A
SCHEMBL10897886 0.80 CES2 (0.67) CES2CES1PARP1NPC1RAB9A
SCHEMBL3198121 0.79 TSHR (0.52) CES2CES1NPC1RAB9AMEN1
SCHEMBL27763784 0.78 MEN1 (0.56) CES2CES1PARP1NPC1RAB9A
SCHEMBL17244237 0.78 CES2 (0.65) CES2CES1PARP1NPC1RAB9A
SCHEMBL30758862 0.78 CES2 (0.69) CES2CES1PARP1NPC1RAB9A
SCHEMBL11248287 0.78 CES2 (0.69) CES2CES1PARP1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0646570-B1 PROCESS FOR PRODUCING LIGNAN COMPOUND SHIONOGI & CO (JP) 1998-06-24 EP disclosed
US-5488134-A Preparation of compounds of lignan series SHIONOGI & CO., LTD. (JP) 1996-01-30 US disclosed
EP-0646570-A1 PROCESS FOR PRODUCING LIGNAN COMPOUND SHIONOGI & CO., LTD. (JP) 1995-04-05 EP disclosed