SCHEMBL8626440

SCHEMBL8626440

COC(=O)C#CC(=O)c1cccc(C)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
PARP1 P09874 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.47
CTNNB1 P35222 1/20 0.47
WNT3A P56704 1/20 0.47
KCNK3 O14649 4/20 0.46
KCNK9 Q9NPC2 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
KCNH2 Q12809 1/20 0.46
RAB9A P51151 3/20 0.46
NPC1 O15118 2/20 0.44
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
POLB P06746 1/20 0.43
TP53 P04637 1/20 0.43
GPR17 Q13304 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8628090 0.82 CES2 (0.59) PARP1SMN1; SMN2KCNK3KCNK9MEN1
SCHEMBL3198121 0.80 TSHR (0.52) SMN1; SMN2MEN1KMT2ARAB9ANPC1
SCHEMBL8627919 0.79 TDP1 (0.53) HDAC6SMN1; SMN2CTNNB1WNT3AMEN1
SCHEMBL27426409 0.78 LOXL2 (0.63) SMN1; SMN2RAB9ANPC1TP53
SCHEMBL10429075 0.78 CTNNB1 (0.48) HDAC8HDAC6PARP1SMN1; SMN2CTNNB1
SCHEMBL29534771 0.74 GPR17 (0.65) HDAC8HDAC6PARP1SMN1; SMN2CTNNB1
SCHEMBL40429 0.74 GPR17 (0.65) HDAC8HDAC6PARP1SMN1; SMN2CTNNB1
SCHEMBL27582425 0.74 PARP1 (0.59) HDAC8HDAC6PARP1SMN1; SMN2KCNK3
SCHEMBL28289702 0.74 GPR17 (0.65) HDAC8HDAC6PARP1SMN1; SMN2CTNNB1
SCHEMBL5512015 0.73 TSHR (0.58) SMN1; SMN2CTNNB1WNT3AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0646570-B1 PROCESS FOR PRODUCING LIGNAN COMPOUND SHIONOGI & CO (JP) 1998-06-24 EP disclosed
US-5488134-A Preparation of compounds of lignan series SHIONOGI & CO., LTD. (JP) 1996-01-30 US disclosed
EP-0646570-A1 PROCESS FOR PRODUCING LIGNAN COMPOUND SHIONOGI & CO., LTD. (JP) 1995-04-05 EP disclosed