SCHEMBL8628472

SCHEMBL8628472

CC(C)(C)OC(=O)NCCCNC(=O)Nc1cccc(C(=O)NCCC(=O)O)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.55
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
PAX8 Q06710 1/20 0.48
SIRT5 Q9NXA8 1/20 0.48
GAA P10253 1/20 0.47
PRMT5 O14744 1/20 0.45
WDR77 Q9BQA1 1/20 0.45
CASR P41180 1/20 0.43
LMNA P02545 1/20 0.43
CCNC P24863 1/20 0.43
CDK8 P49336 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
TP53BP1 Q12888 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8625971 0.88 ALDH1A1 (0.52) EPHX2CA1CA2PAX8GAA
SCHEMBL8628814 0.87 CASR (0.55) EPHX2CA1CA2PAX8CASR
SCHEMBL16152246 0.82 SMN1; SMN2 (0.60) CA1CA2GAASMN1; SMN2TP53BP1
SCHEMBL8623427 0.81 EPHX2 (0.59) EPHX2PAX8GAACASRLMNA
SCHEMBL8897098 0.81 NAMPT (0.56) EPHX2CA1CA2LMNASMN1; SMN2
SCHEMBL31617997 0.81 EPHX1 (0.58) CA1CA2GAALMNACCNC
SCHEMBL30684558 0.81 PPARG (0.51) LMNASMN1; SMN2HDAC3HDAC1HDAC2
SCHEMBL10169791 0.79 CA1 (0.58) CA1CA2PAX8GAACASR
SCHEMBL29459203 0.79 CA1 (0.58) CA1CA2PAX8GAACASR
SCHEMBL284884 0.78 SMN1; SMN2 (0.59) CA1CA2LMNASMN1; SMN2TP53BP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0689549-B1 NEW UREA DERIVATES, THEIR PREPARATION AND THEIR USE HOECHST AG (DE) 1998-06-17 EP disclosed
US-5703050-A INHIBIT PLATELET AGGREGATION, METASTASIS OF CARCINOMA CELLS, OSTEOCLAST BINDING TO BONE SURFACE HOECHST AKTIENGESELLSCHAFT (DE) 1997-12-30 US disclosed
EP-0689549-A1 NEW UREA DERIVATES, THEIR PREPARATION AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1996-01-03 EP disclosed
WO-1994022907-A1 NEW UREA DERIVATES, THEIR PREPARATION AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1994-10-13 WO disclosed