SCHEMBL8628579

SCHEMBL8628579

CC(C)(C)OC(=O)N(CCCCCCCCN(CCCN(Cc1cccc2ccccc12)C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)CCCN(Cc1cccc2ccccc12)C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.46
NR1D1 P20393 1/20 0.44
CYP2D6 P10635 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
MC4R P32245 2/20 0.42
MC5R P33032 2/20 0.42
MC3R P41968 2/20 0.42
MC1R Q01726 2/20 0.42
BACE1 P56817 1/20 0.41
CA14 Q9ULX7 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
ACHE P22303 2/20 0.40
NR1I2 O75469 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21092036 0.87 CYP2D6 (0.45) NPSR1NR1D1CYP2D6CYP1A2CYP2C19
SCHEMBL8021840 0.80 HDAC3 (0.55) CA14CTSSL3MBTL1HDAC1LMNA
SCHEMBL8525848 0.79 HDAC3 (0.56) CA14CTSSL3MBTL1HDAC1LMNA
SCHEMBL13913291 0.77 CA14 (0.43) BACE1CA14L3MBTL1HDAC1LMNA
SCHEMBL3293337 0.77 CA14 (0.41) BACE1CA14L3MBTL1HDAC1ACHE
SCHEMBL27585984 0.77 ADRA2A (0.51) NPSR1NR1D1CYP2D6CYP1A2CYP2C19
SCHEMBL3292650 0.76 CA14 (0.41) BACE1CA14L3MBTL1HDAC1LMNA
SCHEMBL3294768 0.74 SSTR4 (0.40) BACE1CA14L3MBTL1HDAC1LMNA
SCHEMBL1579465 0.74 ADRA2C (0.45) CYP2D6MC3RBACE1HDAC1SLC6A2
SCHEMBL8625900 0.74 L3MBTL1 (0.45) CYP2C19CA14L3MBTL1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753714-A ANTIPROTOZOA AGENTS MERRELL PHARMACEUTICALS INC. (US) 1998-05-19 US disclosed
EP-0277635-A2 Novel polyamine derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-10 EP disclosed