SCHEMBL8628952

SCHEMBL8628952

CSc1ccc(-c2c[nH]nc2-c2ccccc2S(N)(=O)=O)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.41
PTGS1 P23219 4/20 0.41
PTGES2 Q9H7Z7 1/20 0.40
ALOX5AP P20292 4/20 0.35
FEN1 P39748 4/20 0.35
CA2 P00918 3/20 0.34
CA9 Q16790 2/20 0.34
CA1 P00915 2/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RAB9A P51151 1/20 0.34
CA12 O43570 1/20 0.34
TRPV1 Q8NER1 3/20 0.34
F10 P00742 3/20 0.34
F2 P00734 2/20 0.34
PRSS1 P07477 2/20 0.34
CA7 P43166 1/20 0.33
CA13 Q8N1Q1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631083 0.86 PTGES2 (0.53) PTGS2PTGS1PTGES2ALOX5APFEN1
SCHEMBL7779777 0.85 PTGS2 (0.49) PTGS2PTGS1CA2CA9CA1
SCHEMBL8628206 0.83 PTGES2 (0.39) PTGS2PTGES2ALOX5APFEN1CA2
SCHEMBL8631176 0.81 PTGS2 (0.46) PTGS2PTGS1PTGES2CA2CA9
SCHEMBL8627977 0.80 PTGS2 (0.50) PTGS2PTGS1PTGES2CA2CA9
SCHEMBL7779346 0.80 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL8630031 0.79 PTGS2 (0.41) PTGS2PTGS1ALOX5APFEN1CA2
SCHEMBL8631662 0.79 F10 (0.42) PTGES2CA2CA9CA1NPC1
SCHEMBL8628731 0.78 GYS1 (0.47) PTGS2PTGS1ALOX5APFEN1ALDH1A1
SCHEMBL8632840 0.78 LRRK2 (0.42) PTGS2PTGS1CA2CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed