SCHEMBL8629318

SCHEMBL8629318

COc1ccc(-c2c[nH]nc2NS(=O)(=O)c2ccccc2)cc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.50
PTGS1 P23219 3/20 0.50
NR3C1 P04150 1/20 0.47
STAT3 P40763 2/20 0.46
AAK1 Q2M2I8 1/20 0.45
NTRK1 P04629 2/20 0.45
KIT P10721 2/20 0.45
PIK3CA P42336 2/20 0.45
ACLY P53396 3/20 0.44
CDK2 P24941 1/20 0.44
MAPK14 Q16539 1/20 0.43
SCN9A Q15858 1/20 0.43
HTR6 P50406 1/20 0.42
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627771 0.88 ALDH1A1 (0.47) PTGS2PTGS1AAK1NTRK1KIT
SCHEMBL8632810 0.86 STAT3 (0.42) STAT3KITMAPK14SCN9ATUBB4A
SCHEMBL8631045 0.86 STAT3 (0.42) STAT3AAK1PIK3CAACLYMAPK14
SCHEMBL8758715 0.83 ALDH1A1 (0.43) PTGS2PTGS1AAK1NTRK1KIT
SCHEMBL8632208 0.81 STAT3 (0.51) STAT3TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8632663 0.81 CYP17A1 (0.48) NR3C1AAK1PIK3CACDK2MAPK14
SCHEMBL8631178 0.81 STAT3 (0.47) STAT3KITMAPK14
SCHEMBL8635055 0.81 PTGS2 (0.48) PTGS2PTGS1NR3C1STAT3ACLY
SCHEMBL8659801 0.80 STAT3 (0.69) PTGS2PTGS1NR3C1STAT3ACLY
SCHEMBL8630028 0.80 ALDH1A1 (0.45) AAK1NTRK1KITPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed