SCHEMBL8629331

SCHEMBL8629331

CC(CO)C[S+]([O-])c1cnc[nH]1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.35
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
RECQL P46063 1/20 0.34
PMP22 Q01453 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HRH3 Q9Y5N1 5/20 0.34
HRH4 Q9H3N8 4/20 0.34
ALDH1A1 P00352 3/20 0.34
MEN1 O00255 1/20 0.34
GLA P06280 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP1A2 P05177 1/20 0.34
NFKB1 P19838 1/20 0.34
THPO P40225 1/20 0.34
LMNA P02545 1/20 0.33
APEX1 P27695 1/20 0.33
BLM P54132 1/20 0.33
CPB1 P15086 1/20 0.32
CPB2 Q96IY4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4687343 0.84 HRH4 (0.34) HRH3HRH4ALDH1A1MEN1GLA
SCHEMBL22024412 0.70 HRH3 (0.41) PKMHRH3HRH4ALDH1A1MEN1
SCHEMBL4681113 0.68 TRPA1 (0.31)
SCHEMBL15906228 0.67 HRH3 (0.61) PKMKDM4EPOLBRECQLPMP22
SCHEMBL6664741 0.67 HRH3 (0.61) PKMKDM4EPOLBRECQLPMP22
SCHEMBL14390959 0.67 HRH3 (0.61) PKMKDM4EPOLBRECQLPMP22
SCHEMBL4680532 0.67 CHRNB2 (0.34) KDM4ELMNA
SCHEMBL20993530 0.67
SCHEMBL7351528 0.66 TRPA1 (0.32)
SCHEMBL8633118 0.63 PKM (0.37) PKMKDM4EPOLBRECQLPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed