SCHEMBL8629437

SCHEMBL8629437

COc1cccc(C(O)c2scnc2C)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.45
PKM P14618 1/20 0.44
AOC3 Q16853 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
KDM4A O75164 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
IDO1 P14902 1/20 0.40
TDO2 P48775 1/20 0.40
CTSA P10619 1/20 0.40
FGFR2 P21802 1/20 0.39
FGFR4 P22455 1/20 0.39
FGFR3 P22607 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
ALOX5 P09917 1/20 0.38
ACHE P22303 1/20 0.38
CREBBP Q92793 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025658 0.82 IDO1 (0.38) PKMIDO1TDO2CTSAACHE
SCHEMBL8632333 0.81 ADRB1 (0.41) BRD4TSHRACHECREBBP
SCHEMBL8630297 0.81 PFKFB3 (0.38) PKMTSHRALOX5
SCHEMBL8634093 0.80 BRD4 (0.43) BRD4IDO1TDO2ACHECREBBP
SCHEMBL8631276 0.80 BRD4 (0.41) BRD4IDO1TDO2CTSACREBBP
SCHEMBL2593085 0.79 SLC6A3 (0.44) BRD4PKMIDO1TDO2CREBBP
SCHEMBL8631320 0.78 ALDH1A1 (0.37) TSHR
SCHEMBL8656491 0.78 TP53 (0.40) BRD4CREBBP
SCHEMBL9026792 0.77 KMT2A (0.48) L3MBTL1IDO1TDO2KMT2A
SCHEMBL2093768 0.77 AOC3 (0.59) BRD4PKMAOC3L3MBTL1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed