SCHEMBL8629752

SCHEMBL8629752

NS(=O)(=O)c1ccccc1-c1n[nH]cc1-c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA9 Q16790 1/20 0.43
PTGS2 P35354 2/20 0.43
DYRK1A Q13627 1/20 0.41
EDNRA P25101 1/20 0.39
NAMPT P43490 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
STAT3 P40763 1/20 0.38
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
USP2 O75604 1/20 0.37
USP1 O94782 1/20 0.37
USP8 P40818 1/20 0.37
OTUB1 Q96FW1 1/20 0.37
USP36 Q9P275 1/20 0.37
ALOX5AP P20292 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632289 0.86 AKR1B1 (0.40) CA2CA12CA1CA9PTGS2
SCHEMBL8630958 0.85 LRRK2 (0.48) CA2CA1
SCHEMBL5488230 0.83 CA2 (0.56) CA2CA12CA1CA9PTGS2
SCHEMBL7772942 0.83 CA2 (0.62) CA2CA12CA1CA9PTGS2
SCHEMBL8632961 0.80 F10 (0.40) CA2CA12CA1CA9ALOX5AP
SCHEMBL8634768 0.79 F10 (0.42) CA2CA12CA1CA9ALOX5AP
SCHEMBL8627977 0.79 PTGS2 (0.50) CA2CA12CA1CA9PTGS2
SCHEMBL8632840 0.79 LRRK2 (0.42) CA2CA12CA1CA9PTGS2
SCHEMBL8631181 0.79 PTGS2 (0.50) CA9PTGS2ALOX5APFEN1
SCHEMBL8631346 0.79 NPC1 (0.40) CA2CA1DYRK1ANAMPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed