SCHEMBL8630301

SCHEMBL8630301

SC1CCc2ccccc2[N]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
PLAU P00749 1/20 0.36
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
CYP19A1 P11511 3/20 0.34
ADRA1A P35348 1/20 0.34
GRIN2B Q13224 2/20 0.33
IDO1 P14902 2/20 0.33
PDPK1 O15530 1/20 0.33
CYP2D6 P10635 1/20 0.33
MEN1 O00255 1/20 0.33
RECQL P46063 1/20 0.33
KMT2A Q03164 1/20 0.33
ANPEP P15144 1/20 0.32
TSHR P16473 1/20 0.32
CYP17A1 P05093 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1515117 0.77 NOS3 (0.41) NOS3NOS1NOS2PLAUNPC1
SCHEMBL8935522 0.75 CYP2D6 (0.40) NOS3NOS1NOS2PLAUNPC1
SCHEMBL10388003 0.75 NOS3 (0.39) NOS3NOS1NOS2PLAUNPC1
SCHEMBL5542044 0.75 NOS3 (0.39) NOS3NOS1NOS2PLAUNPC1
SCHEMBL11647276 0.69 NOS3 (0.39) NOS3NOS1NOS2NPC1ALDH1A1
SCHEMBL5008486 0.68 NOS3 (0.42) NOS3NOS1NOS2PLAUALDH1A1
SCHEMBL7137711 0.67 HTR1A (0.41) NOS3NOS1NOS2
SCHEMBL6796979 0.66 NOS3 (0.46) NOS3NOS1NOS2MAPTCYP19A1
SCHEMBL688175 0.64 NOS3 (0.56) NOS3NOS1NOS2NPC1ALDH1A1
SCHEMBL6397208 0.62 IDO1 (0.50) IDO1PDPK1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825986-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1998-03-04 EP disclosed
US-5616712-A SKIN DISORDERS; ANTICARCINOGENIC AND -INFLAMMATORY AGENTS; AUTOIMMUNE DISEASES; ALLERGAN (US) 1997-04-01 US disclosed
US-5616712-A SKIN DISORDERS; ANTICARCINOGENIC AND -INFLAMMATORY AGENTS; AUTOIMMUNE DISEASES; ALLERGAN (US) 1997-04-01 US disclosed
WO-1996036609-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-11-21 WO disclosed