SCHEMBL8630356

SCHEMBL8630356

NS(=O)(=O)c1ccccc1-c1nn(Cc2ccccc2)c(C(F)(F)F)c1-c1ccc(Cl)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MARS1 P56192 2/20 0.40
PTGS2 P35354 3/20 0.40
PTGS1 P23219 1/20 0.40
CYP3A4 P08684 3/20 0.37
DPP4 P27487 3/20 0.37
CYP2C19 P33261 3/20 0.37
DPP8 Q6V1X1 2/20 0.37
DPP9 Q86TI2 2/20 0.37
ORAI1 Q96D31 1/20 0.36
CNR1 P21554 1/20 0.36
F10 P00742 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PTGES2 Q9H7Z7 1/20 0.36
TRPV4 Q9HBA0 1/20 0.35
KCNH2 Q12809 1/20 0.35
HSD11B1 P28845 1/20 0.35
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630571 0.89 PTGS2 (0.45) MARS1PTGS2PTGS1DPP4DPP8
SCHEMBL8629984 0.87 PTGS2 (0.44) PTGS2PTGS1CYP3A4CYP2C19F10
SCHEMBL8631997 0.87 PTGS2 (0.39) PTGS2PTGS1F10PTGES2HSD11B1
SCHEMBL8631241 0.86 F10 (0.38) MARS1PTGS2PTGS1F10PTGES2
SCHEMBL7779461 0.86 PTGS2 (0.50) MARS1PTGS2PTGS1MEN1KMT2A
SCHEMBL8627914 0.85 PTGS2 (0.38) PTGS2PTGS1CYP3A4CYP2C19F10
SCHEMBL8630171 0.85 PTGS2 (0.45) PTGS2PTGS1F10MEN1KMT2A
SCHEMBL8631265 0.84 PTGS2 (0.42) PTGS2PTGS1CYP3A4CYP2C19F10
SCHEMBL8632872 0.84 PTGS2 (0.39) PTGS2PTGS1F10ALDH1A1GAA
SCHEMBL8635534 0.81 PTGS2 (0.53) PTGS2PTGS1F10KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed