SCHEMBL8630767

SCHEMBL8630767

COc1cc(N)ccc1C(=O)N1c2ccc(Cl)cc2CCCC1CCOS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 1/20 0.41
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.36
CASP3 P42574 2/20 0.35
CASP7 P55210 2/20 0.35
SCN5A Q14524 1/20 0.35
SCN9A Q15858 1/20 0.35
TP53 P04637 2/20 0.35
DRD2 P14416 1/20 0.35
ALDH1A1 P00352 3/20 0.34
GAA P10253 2/20 0.34
CASP1 P29466 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ACHE P22303 1/20 0.34
HTR4 Q13639 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634668 0.92 AVPR2 (0.51) AVPR2KMT2ACASP3CASP7TP53
SCHEMBL8629507 0.89 KCNMA1 (0.36) POLBKMT2ACASP3CASP7TP53
SCHEMBL8627190 0.89 AVPR2 (0.42) AVPR2POLBKMT2ASCN5ASCN9A
SCHEMBL8634053 0.87 AVPR2 (0.41) AVPR2POLBKMT2ACASP3CASP7
SCHEMBL8630766 0.83 AVPR2 (0.41) AVPR2POLBKMT2ASCN5ASCN9A
SCHEMBL8627187 0.82 AVPR2 (0.40) AVPR2POLBKMT2ASCN5ASCN9A
SCHEMBL8630680 0.82 AVPR2 (0.38) AVPR2KMT2ACASP3CASP7TP53
SCHEMBL4686344 0.80 AVPR2 (0.41) AVPR2CASP3CASP7SCN5ASCN9A
SCHEMBL8633374 0.80 AVPR2 (0.52) AVPR2KMT2ATP53ALDH1A1MAPT
SCHEMBL8630164 0.80 TSHR (0.38) POLBKMT2ATP53ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed