SCHEMBL8630164

SCHEMBL8630164

COc1cc(N)ccc1C(=O)N1c2ccc(F)cc2CCCC1OCCOS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
ALDH1A1 P00352 3/20 0.36
HTT P42858 3/20 0.36
POLB P06746 1/20 0.36
LMNA P02545 1/20 0.36
PDK1 Q15118 7/20 0.36
PDK2 Q15119 7/20 0.36
PDK3 Q15120 7/20 0.36
PDK4 Q16654 7/20 0.36
HSP90AA1 P07900 2/20 0.36
KDM4E B2RXH2 1/20 0.36
TP53 P04637 2/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPT P10636 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627190 0.91 AVPR2 (0.42) POLBTP53KMT2AMAPT
SCHEMBL8634053 0.87 AVPR2 (0.41) POLBTP53KMT2AMAPT
SCHEMBL8630162 0.86 TSHR (0.38) TSHRALDH1A1HTTPOLBLMNA
SCHEMBL8631906 0.85 RORC (0.44) ALDH1A1HTTPOLBLMNAKDM4E
SCHEMBL8633374 0.82 AVPR2 (0.52) ALDH1A1HTTLMNAPDK1PDK2
SCHEMBL4686263 0.81 HTR4 (0.34) TSHRALDH1A1POLBKDM4EMEN1
SCHEMBL8627538 0.80 KCNMA1 (0.36) ALDH1A1HTTPOLBLMNATP53
SCHEMBL8630767 0.80 AVPR2 (0.41) TSHRALDH1A1POLBTP53KMT2A
SCHEMBL8629474 0.78 AVPR2 (0.51) LMNAPDK1PDK2PDK3PDK4
SCHEMBL8630395 0.78 PDK1 (0.35) TSHRALDH1A1HTTLMNAPDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed