SCHEMBL8630808

SCHEMBL8630808

Cc1cc(C(=O)NP(N)(N)=O)c(C)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
BACE1 P56817 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 2/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PLA2G10 O15496 2/20 0.36
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
ALOX5 P09917 1/20 0.35
TSHR P16473 1/20 0.34
CTSV O60911 1/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
PSMD14 O00487 1/20 0.33
MMP2 P08253 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634456 0.84 MAPT (0.41) NPC1RAB9AALDH1A1MAPTGAA
SCHEMBL8628998 0.83 MAPT (0.43) NPC1RAB9AALDH1A1MAPTL3MBTL1
SCHEMBL8587274 0.75 CCNB2 (0.33) NPC1RAB9AALDH1A1MAPTGAA
SCHEMBL17367390 0.72 PLA2G10 (0.49) NPC1RAB9AALDH1A1MAPTGAA
SCHEMBL11848005 0.72 ALDH1A1 (0.44) NPC1RAB9AALDH1A1MAPTGAA
SCHEMBL2996683 0.72 ALDH1A1 (0.44) NPC1RAB9AALDH1A1MAPTGAA
SCHEMBL8630712 0.71 NAMPT (0.47) NPC1RAB9AALDH1A1MAPTGAA
SCHEMBL8636004 0.70 ALDH1A1 (0.49) NPC1RAB9AALDH1A1MAPTLMNA
SCHEMBL15296667 0.70 NPC1 (0.40) NPC1RAB9APLA2G10
SCHEMBL248005 0.70 SMN1; SMN2 (0.43) NPC1RAB9AALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840917-A ADMINISTERING TO MAMMAL TO ERADICATE HELICOBACTER PYLORI TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-24 US disclosed
EP-0852498-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-07-15 EP disclosed
WO-1997011705-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-03 WO disclosed