SCHEMBL8631055

SCHEMBL8631055

CCn1[c]nnc1-c1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
ALDH1A1 P00352 7/20 0.44
CYP2A6 P11509 3/20 0.44
CYP3A4 P08684 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
CYP2E1 P05181 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44
LMNA P02545 4/20 0.44
KDM4E B2RXH2 3/20 0.44
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
HTT P42858 3/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 2/20 0.42
TP53 P04637 1/20 0.42
ALOX15 P16050 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629015 0.88 LMNA (0.43) CYP2C19CYP1A2TDP1ALDH1A1CYP2A6
SCHEMBL794659 0.82 TSHR (0.43) ALDH1A1KDM4EHPGDSMN1; SMN2HSD17B10
SCHEMBL8629217 0.79 ALDH1A1 (0.47) CYP2C19CYP1A2ALDH1A1CYP2A6CYP3A4
SCHEMBL8682578 0.72 HIF1A (0.48) CYP2C19TDP1ALDH1A1CYP3A4CYP2C9
SCHEMBL26970988 0.71 ALDH1A1 (0.59) CYP2C19CYP1A2TDP1ALDH1A1CYP2A6
SCHEMBL18104668 0.70 ALDH1A1 (0.58) CYP2C19CYP1A2TDP1ALDH1A1CYP2A6
SCHEMBL1545128 0.69 ALDH1A1 (0.56) CYP2C19CYP1A2TDP1ALDH1A1CYP2A6
SCHEMBL28429543 0.66 KMT2A (0.61) CYP1A2TDP1ALDH1A1CYP2A6CYP3A4
SCHEMBL22046643 0.66 ALDH1A1 (0.74) ALDH1A1L3MBTL1LMNAKDM4EHTT
SCHEMBL30522532 0.66 TBXAS1 (0.45) CYP2C19CYP1A2TDP1ALDH1A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35754-E FOR TREATING BACTERIAL INFECTIONS HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
US-5710146-A ANTIBIOTICS FOR BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4399131-A Cephem derivatives HOECHST AG (DE) 1983-08-16 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed