SCHEMBL8631273

SCHEMBL8631273

Cc1ncsc1C(O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.41
SLC6A2 P23975 8/20 0.39
SLC6A4 P31645 8/20 0.39
SLC6A3 Q01959 8/20 0.39
CYP3A4 P08684 6/20 0.35
CYP2D6 P10635 6/20 0.35
PTPN5 P54829 3/20 0.35
KCNH2 Q12809 5/20 0.34
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
S1PR2 O95136 1/20 0.33
S1PR4 O95977 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634063 0.83 FFAR2 (0.38) BRD4ALDH1A1LMNA
SCHEMBL8631276 0.81 BRD4 (0.41) BRD4SLC6A3CYP3A4KCNH2
SCHEMBL9026067 0.79 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL9025658 0.77 IDO1 (0.38) SLC6A3LMNA
SCHEMBL9026742 0.76 ATM (0.38) BRD4SLC6A2SLC6A3
SCHEMBL8683323 0.76 KDM4E (0.43) SLC6A3CYP2D6ALDH1A1LMNA
SCHEMBL8630297 0.76 PFKFB3 (0.38) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL8632333 0.76 ADRB1 (0.41) BRD4SLC6A3LMNA
SCHEMBL2593085 0.76 SLC6A3 (0.44) BRD4SLC6A3ALDH1A1LMNAHTT
SCHEMBL8633346 0.75 LMNA (0.40) LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed