SCHEMBL8631977

SCHEMBL8631977

CC(=O)C(Oc1cccc(C)c1)C(=O)ON1CCN(c2ccncc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.42
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
MAPT P10636 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
AOC3 Q16853 2/20 0.39
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TSHR P16473 4/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HRH3 Q9Y5N1 2/20 0.37
GFER P55789 1/20 0.37
GAA P10253 1/20 0.37
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
LMNA P02545 2/20 0.36
MAPK1 P28482 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630734 0.89 ROCK2 (0.52) ROCK2ITGB3ITGA2BMAPTAOC3
SCHEMBL8633669 0.89 CYP2C9 (0.44) ROCK2ITGB3ITGA2BMAPTALDH1A1
SCHEMBL8636239 0.82 CHRM1 (0.39) ROCK2ITGB3ITGA2BAOC3ALDH1A1
SCHEMBL8634919 0.82 CYP2C9 (0.37) ROCK2ITGB3ITGA2BMAPTAOC3
SCHEMBL8633528 0.80 AOC3 (0.39) MAPTKMT2AAOC3ALDH1A1TSHR
SCHEMBL8634776 0.80 AOC3 (0.38) ROCK2ITGB3ITGA2BMAPTAOC3
SCHEMBL8632221 0.80 TSHR (0.40) ROCK2ITGB3ITGA2BMAPTMEN1
SCHEMBL8632788 0.78 MAPT (0.37) MAPTKMT2AALDH1A1KDM4ETSHR
SCHEMBL8632956 0.74 CYP2C9 (0.38) ROCK2ITGB3ITGA2BMAPTALDH1A1
Hydrochloric Acid SCHEMBL8681516 0.73 CYP2C9 (0.38) ROCK2ITGB3ITGA2BMAPTAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed