SCHEMBL8636239

SCHEMBL8636239

CC(=O)C(Oc1c(Cl)cccc1Cl)C(=O)ON1CCN(c2ccncc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.39
AOC3 Q16853 2/20 0.37
AKR1C3 P42330 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
ROCK2 O75116 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
HTR4 Q13639 1/20 0.36
HRH3 Q9Y5N1 2/20 0.35
HIF1A Q16665 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
LSS P48449 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634776 0.85 AOC3 (0.38) AOC3CYP2C9TSHRROCK2ITGB3
SCHEMBL8633669 0.83 CYP2C9 (0.44) CYP2C9TSHRROCK2ITGB3ITGA2B
SCHEMBL8630734 0.82 ROCK2 (0.52) AOC3ROCK2ITGB3ITGA2BALDH1A1
SCHEMBL8631977 0.82 ROCK2 (0.42) AOC3CYP2C9TSHRROCK2ITGB3
SCHEMBL8632221 0.80 TSHR (0.40) AOC3CYP2C9TSHRROCK2ITGB3
SCHEMBL8634919 0.80 CYP2C9 (0.37) AOC3CYP2C9TSHRROCK2ITGB3
SCHEMBL8699531 0.73 ADRB2 (0.41) CYP2C9TSHRITGB3ITGA2BHRH3
SCHEMBL8838126 0.73 CYP2C9 (0.51) AKR1C3CYP2C9TSHRTRPV1ITGB3
Hydrochloric Acid SCHEMBL8838111 0.71 CYP2C9 (0.50) AOC3AKR1C3CYP2C9TSHRTRPV1
Hydrochloric Acid SCHEMBL8838033 0.71 CYP2C9 (0.50) AOC3AKR1C3CYP2C9TSHRTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed