SCHEMBL8634776

SCHEMBL8634776

CC(=O)C(Oc1c(C(C)(C)C)cccc1C(C)(C)C)C(=O)ON1CCN(c2ccncc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.38
ROCK2 O75116 1/20 0.36
CYP2C9 P11712 2/20 0.36
TSHR P16473 1/20 0.36
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
GAA P10253 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
HRH3 Q9Y5N1 5/20 0.34
P2RY1 P47900 2/20 0.34
HIF1A Q16665 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PLOD2 O00469 1/20 0.34
PLOD3 O60568 1/20 0.34
PLOD1 Q02809 1/20 0.34
SPHK1 Q9NYA1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8636239 0.85 CHRM1 (0.39) AOC3ROCK2CYP2C9TSHRITGB3
SCHEMBL8633669 0.81 CYP2C9 (0.44) ROCK2CYP2C9TSHRITGB3ITGA2B
SCHEMBL8630734 0.80 ROCK2 (0.52) AOC3ROCK2ITGB3ITGA2BGAA
SCHEMBL8631977 0.80 ROCK2 (0.42) AOC3ROCK2CYP2C9TSHRITGB3
SCHEMBL8632221 0.79 TSHR (0.40) AOC3ROCK2CYP2C9TSHRITGB3
SCHEMBL8634919 0.79 CYP2C9 (0.37) AOC3ROCK2CYP2C9TSHRITGB3
SCHEMBL8699531 0.72 ADRB2 (0.41) CYP2C9TSHRITGB3ITGA2BGAA
SCHEMBL8838126 0.71 CYP2C9 (0.51) CYP2C9TSHRITGB3ITGA2BGAA
SCHEMBL8634772 0.70 GAA (0.39) AOC3ROCK2CYP2C9TSHRITGB3
Hydrochloric Acid SCHEMBL8838111 0.70 CYP2C9 (0.50) AOC3CYP2C9TSHRITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed