SCHEMBL8632229

SCHEMBL8632229

CN(C)C1CCC(Cl)N(C(=O)c2ccc(NC(=O)c3ccccc3Cl)cc2)c2ccc(O)cc21

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 5/20 0.47
AVPR2 P30518 3/20 0.47
AVPR1B P47901 3/20 0.47
CHRM1 P11229 2/20 0.47
ABCB11 O95342 1/20 0.47
HTR1A P08908 1/20 0.47
OXTR P30559 1/20 0.47
SLC6A4 P31645 1/20 0.47
ADRA1A P35348 1/20 0.47
OPRM1 P35372 1/20 0.47
HSD11B1 P28845 1/20 0.45
SMO Q99835 1/20 0.40
CHRM5 P08912 1/20 0.40
CHRM3 P20309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8717630 0.90 AVPR1A (0.57) AVPR1AAVPR2AVPR1BCHRM1ABCB11
SCHEMBL8628412 0.88 AVPR1A (0.44) AVPR1AAVPR2AVPR1BCHRM1ABCB11
SCHEMBL8628393 0.85 AVPR2 (0.42) AVPR1AAVPR2AVPR1BCHRM1ABCB11
SCHEMBL8716136 0.82 AVPR1A (0.47) AVPR1AAVPR2AVPR1BCHRM1ABCB11
SCHEMBL8712963 0.81 AVPR1A (0.69) AVPR1AAVPR2AVPR1BCHRM1ABCB11
SCHEMBL8714659 0.81 AVPR1A (0.57) AVPR1AAVPR2AVPR1BCHRM1ABCB11
SCHEMBL8718316 0.80 AVPR1A (0.56) AVPR1AAVPR2AVPR1BCHRM1ABCB11
SCHEMBL8712973 0.79 AVPR1A (0.54) AVPR1AAVPR2AVPR1BCHRM1ABCB11
SCHEMBL8717780 0.79 AVPR1A (0.54) AVPR1AAVPR2AVPR1BCHRM1ABCB11
SCHEMBL8713819 0.78 HSD11B1 (0.49) AVPR1AAVPR2AVPR1BHSD11B1SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed