SCHEMBL8716136

SCHEMBL8716136

CCN(C)C1CCC(Cl)N(C(=O)c2ccc(NC(=O)c3ccccc3Cl)cc2)c2ccccc21

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 3/20 0.47
AVPR1B P47901 2/20 0.47
AVPR2 P30518 2/20 0.47
ABCB11 O95342 1/20 0.47
HTR1A P08908 1/20 0.47
CHRM1 P11229 1/20 0.47
OXTR P30559 1/20 0.47
SLC6A4 P31645 1/20 0.47
ADRA1A P35348 1/20 0.47
OPRM1 P35372 1/20 0.47
HSD11B1 P28845 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8717630 0.91 AVPR1A (0.57) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL8713819 0.83 HSD11B1 (0.49) AVPR1AAVPR1BAVPR2HSD11B1
SCHEMBL8712963 0.82 AVPR1A (0.69) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL8714659 0.82 AVPR1A (0.57) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL8632229 0.82 AVPR1A (0.47) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL8715966 0.81 AVPR1A (0.55) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL8718316 0.81 AVPR1A (0.56) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL8713384 0.80 HSD11B1 (0.48) AVPR1AAVPR1BAVPR2HSD11B1
SCHEMBL8717780 0.80 AVPR1A (0.54) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL8712973 0.80 AVPR1A (0.54) AVPR1AAVPR1BAVPR2ABCB11HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753677-A Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed