SCHEMBL8632343

SCHEMBL8632343

CSc1cc(Br)ccc1C(N)=CC(=O)C1CC1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.35
LSS P48449 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
RAB9A P51151 2/20 0.31
AR P10275 1/20 0.31
ATM Q13315 1/20 0.31
MAPT P10636 2/20 0.31
SIRT1 Q96EB6 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30
ABL1 P00519 1/20 0.30
NPC1 O15118 1/20 0.30
AAK1 Q2M2I8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632340 1.00 DGAT1 (0.35) DGAT1LSSSMN1; SMN2RAB9AAR
SCHEMBL8629066 0.84 ADRA1D (0.34) SMN1; SMN2RAB9AMAPTKDM4EMEN1
SCHEMBL8629068 0.84 ADRA1D (0.34) SMN1; SMN2RAB9AMAPTKDM4EMEN1
SCHEMBL8632344 0.83 DGAT1 (0.38) DGAT1SMN1; SMN2RAB9AATMMAPT
SCHEMBL8630195 0.81 SLC6A9 (0.38) MAPTKDM4EGAAHPGD
SCHEMBL8630198 0.81 SLC6A9 (0.38) MAPTKDM4EGAAHPGD
SCHEMBL8631720 0.76 ERN1 (0.33)
SCHEMBL8631716 0.76 ERN1 (0.33)
SCHEMBL8650089 0.76 HPGD (0.36) SMN1; SMN2RAB9AMAPTKDM4EHPGD
SCHEMBL8650094 0.76 HPGD (0.36) SMN1; SMN2RAB9AMAPTKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705243-B1 BETA-AMINOVINYL KETONES, PREPARATION METHOD THEREFOR AND USE THEREOF FOR PREPARING BETA DIKETONES RHONE POULENC AGROCHIMIE (FR) 1998-06-24 EP disclosed
US-5684206-A CONDENSING METHYL ORGANO KETONE WITH A BENZONITRILE IN PRESENCE OF STRONG BASE RHONE-POULENC ARGOCHIMIE (FR) 1997-11-04 US disclosed
EP-0705243-A1 BETA-AMINOVINYL KETONES, PREPARATION METHOD THEREFOR AND USE THEREOF FOR PREPARING BETA DIKETONES RHONE-POULENC AGROCHIMIE (FR) 1996-04-10 EP disclosed
WO-1995000476-A1 BETA-AMINOVINYL KETONES, PREPARATION METHOD THEREFOR AND USE THEREOF FOR PREPARING BETA DIKETONES RHONE POULENC AGROCHIMIE (FR) 1995-01-05 WO disclosed