SCHEMBL8632726

SCHEMBL8632726

CCN(Cc1ccccc1)N1CCN(c2ccncc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KHK P50053 4/20 0.44
CHRNA7 P36544 1/20 0.44
DRD4 P21917 2/20 0.43
HRH1 P35367 2/20 0.43
HRH3 Q9Y5N1 2/20 0.43
CHKA P35790 1/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
RORC P51449 1/20 0.40
HRH2 P25021 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12261943 0.74 DRD4 (0.77) DRD4HRH1HRH3
SCHEMBL3440293 0.73 HRH1 (0.52) HRH1HRH3MAPTHRH2
SCHEMBL18590696 0.73 CHKA (0.67) KHKCHRNA7DRD4HRH1HRH3
SCHEMBL4712908 0.70 CHRNA7 (0.66) CHRNA7HRH3CHKAKDM4EGAA
SCHEMBL28112415 0.69 CHKA (0.80) CHKAKDM4EGAAMAPT
SCHEMBL786054 0.69 ACHE (0.47)
SCHEMBL785872 0.69 ACHE (0.46) HRH1HRH3CHKARORC
SCHEMBL1669246 0.68 DRD4 (0.77) KHKDRD4KDM4E
SCHEMBL14248010 0.67 LMNA (0.73) CHKAKDM4EMAPT
SCHEMBL8251460 0.66 POLB (0.56) DRD4CHKAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed