SCHEMBL8632791

SCHEMBL8632791

CCCCS(=O)(=O)N(C)c1ccc(C(=O)CBr)cc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 8/20 0.44
THRA P10827 3/20 0.41
THRB P10828 2/20 0.41
PTPN1 P18031 5/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
GALR3 O60755 1/20 0.41
RAB9A P51151 1/20 0.41
CNR2 P34972 1/20 0.39
HSD17B3 P37058 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
STS P08842 1/20 0.37
REV1 Q9UBZ9 1/20 0.37
HTR7 P34969 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6301951 0.79 ESR1 (0.44) KDM4ENPC1GALR3RAB9ACNR2
SCHEMBL12352208 0.76 CNR2 (0.47) THRATHRBKDM4ENPC1GALR3
SCHEMBL8910873 0.75 CA12 (0.43) KDM4ENPC1RAB9ACNR2
SCHEMBL1830052 0.73 ESR1 (0.47) KDM4ECNR2HSD17B3
SCHEMBL7182118 0.73 ESR1 (0.47) KDM4ECNR2HSD17B3
SCHEMBL7404753 0.72 THRA (0.62) GSK3BTHRAPTPN1KDM4E
SCHEMBL774179 0.72 GSK3B (0.61) GSK3BPTPN1KDM4ENPC1RAB9A
SCHEMBL10001068 0.72 GSK3B (0.61) GSK3BPTPN1KDM4ENPC1RAB9A
SCHEMBL10001066 0.72 GSK3B (0.61) GSK3BPTPN1KDM4ENPC1RAB9A
SCHEMBL1006322 0.72 GSK3B (0.55) GSK3BTHRATHRBPTPN1HSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed