SCHEMBL1006322

SCHEMBL1006322

CC(C)N(c1ccc(C(=O)CBr)cc1)C(C)C

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 11/20 0.55
PTPN1 P18031 6/20 0.52
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
ABCB1 P08183 1/20 0.37
HSD17B3 P37058 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
USP5 P45974 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10001066 0.79 GSK3B (0.61) GSK3BPTPN1HDAC1HDAC6
SCHEMBL774179 0.79 GSK3B (0.61) GSK3BPTPN1HDAC1HDAC6
SCHEMBL10001068 0.79 GSK3B (0.61) GSK3BPTPN1HDAC1HDAC6
SCHEMBL2497217 0.78 HPGD (0.58) ABCB1
SCHEMBL205280 0.77 GSK3B (0.80) GSK3BPTPN1HDAC3HDAC4HDAC1
SCHEMBL925065 0.76 TSHR (0.52)
SCHEMBL483963 0.76 GSK3B (0.57) GSK3BPTPN1HDAC3HDAC4HDAC1
SCHEMBL182091 0.75 USP5 (0.61) GSK3BPTPN1USP5
SCHEMBL1128718 0.75 PARP10 (0.50)
SCHEMBL960521 0.74 MPO (0.52) HDAC3HDAC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120165227-A1 COMPOUNDS AND METHODS FOR DETECTION AND QUANTIFICATION OF CARBOXYLIC ACIDS THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2012-06-28 US disclosed
WO-2011003193-A1 COMPOUNDS AND METHODS FOR DETECTION AND QUANTIFICATION OF CARBOXYLIC ACIDS THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2011-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120165227-A1 COMPOUNDS AND METHODS FOR DETECTION AND QUANTIFICATION OF CARBOXYLIC ACIDS AKR1C3, AR, AKR1C4 GSK3B 4527/4885PTPN1 4590/4885THRA 1081/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.