SCHEMBL8632808

SCHEMBL8632808

CCOC(=O)c1n[c]sc1N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 0.49
CYP1A2 P05177 2/20 0.49
MAPT P10636 9/20 0.49
HPGD P15428 8/20 0.49
GAA P10253 5/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
FHIT P49789 1/20 0.45
KMT2A Q03164 4/20 0.42
HSD17B10 Q99714 4/20 0.42
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
MEN1 O00255 3/20 0.41
MAPK1 P28482 2/20 0.41
ALOX15 P16050 2/20 0.41
KDM4E B2RXH2 2/20 0.40
APP P05067 1/20 0.40
LMNA P02545 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAOA P21397 1/20 0.40
GRM6 O15303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7236189 0.82 ALDH1A1 (0.44) ALDH1A1CYP1A2MAPTHPGDGAA
SCHEMBL9842107 0.81 ALDH1A1 (0.50) ALDH1A1CYP1A2MAPTHPGDGAA
SCHEMBL27855619 0.79 ALDH1A1 (0.41) ALDH1A1CYP1A2MAPTHPGDGAA
SCHEMBL27855697 0.79 ALDH1A1 (0.41) ALDH1A1CYP1A2MAPTHPGDGAA
SCHEMBL2442977 0.76 LMNA (0.49) ALDH1A1CYP1A2MAPTHPGDGAA
SCHEMBL971952 0.71 ALDH1A1 (0.44) ALDH1A1CYP1A2MAPTHPGDGAA
SCHEMBL2843820 0.71 ALDH1A1 (0.59) ALDH1A1CYP1A2MAPTHPGDGAA
SCHEMBL7516781 0.70 TSHR (0.58) ALDH1A1CYP1A2MAPTHPGDGAA
SCHEMBL1194383 0.70 ALDH1A1 (0.58) ALDH1A1CYP1A2MAPTHPGDGAA
SCHEMBL2367363 0.69 ALDH1A1 (0.57) ALDH1A1CYP1A2MAPTHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35754-E FOR TREATING BACTERIAL INFECTIONS HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
US-5710146-A ANTIBIOTICS FOR BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4399131-A Cephem derivatives HOECHST AG (DE) 1983-08-16 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed