SCHEMBL8633263

SCHEMBL8633263

COc1ccc(N2CCN(Cc3nn(C(C)=O)c4cc(F)ccc34)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.48
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
MAPT P10636 4/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
LMNA P02545 3/20 0.46
ALDH1A1 P00352 3/20 0.45
TRPV4 Q9HBA0 1/20 0.44
HTT P42858 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PAX8 Q06710 1/20 0.43
MAPK1 P28482 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HTR7 P34969 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797687 0.81 KDM4E (0.49) SMOMEN1KMT2AL3MBTL1LMNA
SCHEMBL9393050 0.77 ALDH1A1 (0.45) SMOMEN1KMT2AMAPTL3MBTL1
SCHEMBL8629937 0.75 MAPT (0.53) SMOMEN1KMT2AMAPTL3MBTL1
SCHEMBL8864058 0.73 MEN1 (0.44) MEN1KMT2AALDH1A1MAPK1HTR7
SCHEMBL8631068 0.71 PDGFRA (0.46) MEN1KMT2AKDM4E
SCHEMBL28313258 0.70 MAPT (0.68) SMOMEN1KMT2AMAPTL3MBTL1
Oxalic Acid SCHEMBL10640941 0.67 KDM4E (0.49) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL8630130 0.67 MAPT (0.47) SMOMEN1KMT2AMAPTL3MBTL1
SCHEMBL20291632 0.66 KDM4E (0.58) SMOMEN1KMT2AMAPTL3MBTL1
SCHEMBL8303856 0.65 PDGFRA (0.47) LMNAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780475-A Antipsychotic indazole derivatives MERCK, SHARP & DOHME LIMITED (GB) 1998-07-14 US disclosed
EP-0689539-B1 ANTIPSYCHOTIC INDAZOLE DERIVATIVES MERCK SHARP & DOHME (GB) 1997-12-03 EP disclosed
WO-1994021630-A1 ANTIPSYCHOTIC INDAZOLE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1994-09-29 WO disclosed