SCHEMBL8633503

SCHEMBL8633503

CC1C(c2ccccc2)N(c2ccncc2)CCN1C(CCC(=O)O)Oc1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ITGB3 P05106 3/20 0.33
ITGA2B P08514 3/20 0.33
CYP2C9 P11712 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MAPK1 P28482 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32
HIF1A Q16665 1/20 0.32
DGAT2 Q96PD7 1/20 0.32
SMO Q99835 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
ADAMTS5 Q9UNA0 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632567 0.80 GFER (0.39) MAPTNPSR1ITGB3ITGA2BCYP2C9
SCHEMBL7450096 0.80 ITGB3 (0.42) ITGB3ITGA2BCYP2C9SMN1; SMN2MAPK1
SCHEMBL8636934 0.79 MAPT (0.36) MAPTNPSR1ITGB3ITGA2BCYP2C9
Hydrochloric Acid SCHEMBL8637210 0.79 GFER (0.38) MAPTNPSR1ITGB3ITGA2BMAPK1
SCHEMBL7398021 0.75 ITGB3 (0.39) ITGB3ITGA2BCYP2C9SMN1; SMN2MAPK1
SCHEMBL7403452 0.73 ITGB3 (0.37) ITGB3ITGA2BCYP2C9SMN1; SMN2MAPK1
SCHEMBL8634865 0.72 GAA (0.38) MAPTNPSR1MEN1KMT2ATSHR
SCHEMBL8698839 0.70 FAAH (0.37) NPSR1ITGB3ITGA2BCYP2C9SMN1; SMN2
SCHEMBL8637925 0.70 GFER (0.38) MAPK1ALDH1A1TSHRADAMTS5MMP2
SCHEMBL8630686 0.70 ITGB3 (0.37) ITGB3ITGA2BCYP2C9SMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed