SCHEMBL8634865

SCHEMBL8634865

COC(=O)CCC(Oc1ccccc1)N1CCN(c2ccncc2)C(c2ccccc2)C1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ADAM17 P78536 1/20 0.35
LMNA P02545 1/20 0.34
ROCK2 O75116 2/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KDM1A O60341 1/20 0.33
PRKG1 Q13976 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MEN1 O00255 1/20 0.32
GFER P55789 1/20 0.32
KMT2A Q03164 1/20 0.32
TSHR P16473 1/20 0.32
BUB1 O43683 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8636934 0.90 MAPT (0.36) GAAL3MBTL1MAPTNPSR1ADAM17
SCHEMBL8632567 0.79 GFER (0.39) MAPTNPSR1ROCK2PRKG1GFER
SCHEMBL8637925 0.79 GFER (0.38) GAANPC1RAB9AGFERTSHR
Hydrochloric Acid SCHEMBL8637210 0.79 GFER (0.38) MAPTNPSR1ROCK2PRKG1GFER
SCHEMBL8632725 0.76 ALDH1A1 (0.36) GAAL3MBTL1NPSR1
SCHEMBL8697195 0.74 ROCK2 (0.38) GAANPSR1ROCK2TSHR
SCHEMBL27442362 0.73 GAA (0.43) GAAMAPTNPSR1ROCK2TSHR
SCHEMBL8633503 0.72 MAPT (0.34) MAPTNPSR1MEN1GFERKMT2A
SCHEMBL8633129 0.69 KDM4D (0.35) GAAL3MBTL1NPSR1ROCK2KMT2A
SCHEMBL8686282 0.68 ROCK2 (0.35) ROCK2PRKG1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed