SCHEMBL8633969

SCHEMBL8633969

CCc1cc(Nc2ccc(Cl)cc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.43
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
IDH1 O75874 3/20 0.38
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
F10 P00742 1/20 0.37
CCR2 P41597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635300 0.89 HTT (0.38) MAPTPTGS1PTGS2
SCHEMBL8635140 0.89 BCAT2 (0.42) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL8633209 0.87 MEN1 (0.43) CNR2MEN1KMT2AAKR1C3AKR1C2
SCHEMBL8634230 0.87 AKR1C3 (0.45) MEN1KMT2AAKR1C3AKR1C2LMNA
SCHEMBL8634502 0.86 PTGS1 (0.38) KMT2ACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL7764117 0.86 AKR1C3 (0.42) CNR2MEN1KMT2ACYP3A4CYP2D6
SCHEMBL8635360 0.86 TBXA2R (0.41) LMNAPOLB
SCHEMBL27349234 0.86 RAPGEF4 (0.40) MEN1KMT2ACYP1A2POLBMAPT
SCHEMBL8631102 0.85 AKR1C3 (0.47) CNR2FLT1FLT4KDRMEN1
SCHEMBL7765594 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057999-C 4-Aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed
CN-1138575-A 4-aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-12-25 CN disclosed