SCHEMBL8635262

SCHEMBL8635262

CC(=O)N(C(=O)COc1ccccc1)N1CCN(c2ccncc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
HRH3 Q9Y5N1 7/20 0.47
MAPK1 P28482 3/20 0.47
HRH1 P35367 3/20 0.46
HRH2 P25021 1/20 0.46
ME2 P23368 1/20 0.46
ME1 P48163 1/20 0.46
ME3 Q16798 1/20 0.46
KDM4E B2RXH2 2/20 0.44
TSHR P16473 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HIF1A Q16665 1/20 0.44
HSD17B10 Q99714 1/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696504 0.76 HRH3 (0.51) ITGB3ITGA2BHRH3MAPK1HRH1
SCHEMBL8630427 0.73 ITGB3 (0.47) ITGB3ITGA2BHRH3MAPK1HRH1
SCHEMBL8634854 0.72 ITGB3 (0.51) ITGB3ITGA2BHRH3MAPK1HRH1
SCHEMBL8634182 0.70 HRH3 (0.65) ITGB3ITGA2BHRH3HRH1HRH2
SCHEMBL8695771 0.70 KCNH2 (0.43) ITGB3ITGA2BHRH3MAPK1HRH1
SCHEMBL8634890 0.70 HRH3 (0.50) ITGB3ITGA2BHRH3MAPK1HRH1
SCHEMBL4384247 0.69 HRH3 (0.66) HRH3MAPK1ME2ME1ME3
SCHEMBL8654423 0.69 ITGB3 (0.45) ITGB3ITGA2BHRH3MAPK1HRH1
SCHEMBL4377632 0.68 MAPK1 (0.75) MAPK1KDM4ETSHRNPSR1ALDH1A1
SCHEMBL13636355 0.68 HRH3 (0.65) ITGB3ITGA2BHRH3MAPK1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed