SCHEMBL8635320

SCHEMBL8635320

O=C(Cl)OCOCc1cccnc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.51
CYP17A1 P05093 1/20 0.50
CYP19A1 P11511 1/20 0.50
NAPRT Q6XQN6 1/20 0.47
KMT2A Q03164 3/20 0.47
ALDH1A1 P00352 3/20 0.47
LMNA P02545 2/20 0.47
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
HDAC1 Q13547 1/20 0.43
RECQL P46063 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
GRM5 P41594 1/20 0.43
NAMPT P43490 1/20 0.42
TBXAS1 P24557 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL445196 0.87 ALDH1A1 (0.61) HSD11B1CYP17A1CYP19A1NAPRTKMT2A
Hydrochloric Acid SCHEMBL28059160 0.85 ALDH1A1 (0.59) HSD11B1CYP17A1CYP19A1NAPRTKMT2A
SCHEMBL13630753 0.81 CYP1A2 (0.52) HSD11B1NAPRTTDP1CYP1A2CHRM2
SCHEMBL8454471 0.80 ALDH1A1 (0.71) KMT2AALDH1A1LMNATDP1
SCHEMBL774727 0.80 HSD11B1 (0.44) HSD11B1CYP17A1CYP19A1NAPRTKMT2A
SCHEMBL29563668 0.77 LMNA (0.51) HSD11B1CYP17A1CYP19A1NAPRTKMT2A
SCHEMBL493020 0.77 CYP1A2 (0.56) HSD11B1NAPRTTDP1CYP1A2CHRM2
SCHEMBL4245622 0.76 KMT2A (0.58) HSD11B1CYP17A1CYP19A1NAPRTKMT2A
SCHEMBL28711108 0.76 KMT2A (0.58) CYP17A1CYP19A1NAPRTKMT2AALDH1A1
SCHEMBL361358 0.76 NAPRT (0.61) HSD11B1CYP17A1CYP19A1NAPRTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5789595-A ANTICOAGULANTS TERUMO KABUSHIKI KAISHA (JP) 1998-08-04 US disclosed
EP-0790247-A1 TETRAHYDROISOQUINOLINE DERIVATIVE AND MEDICINAL PREPARATION CONTAINING THE SAME TERUMO KABUSHIKI KAISHA (JP) 1997-08-20 EP disclosed