SCHEMBL8635359

SCHEMBL8635359

O=C(CCNC(=O)c1ccccc1)ON1CCN(c2ccncc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.51
CTSG P08311 1/20 0.51
CTRB1 P17538 1/20 0.51
CMA1 P23946 1/20 0.51
KDM4E B2RXH2 1/20 0.50
HTT P42858 1/20 0.50
DRD2 P14416 2/20 0.49
HTR1A P08908 1/20 0.48
HTR2A P28223 1/20 0.48
DRD3 P35462 1/20 0.48
DRD4 P21917 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7501490 0.81 DRD2 (0.56) DRD2HTR1ADRD3
SCHEMBL7402710 0.79 DRD2 (0.59) DRD2
Hydrochloric Acid SCHEMBL27908881 0.79 DRD2 (0.72) DRD2
SCHEMBL7501496 0.79 PLOD2 (0.56) DRD2DRD4
SCHEMBL8837938 0.79 CHKA (0.47)
SCHEMBL8635423 0.78 F10 (0.52) PRSS1
SCHEMBL2355678 0.78 DRD3 (0.72) DRD2HTR1AHTR2ADRD3DRD4
SCHEMBL8631458 0.78 HRH3 (0.50) KDM4E
SCHEMBL8837943 0.78 ITGB3 (0.48)
Hydrochloric Acid SCHEMBL8838098 0.77 CHKA (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed