SCHEMBL8635498

SCHEMBL8635498

COc1cc(-n2c(C)nc3cccc(C(=O)O)c32)ccc1-c1ccccc1-c1nnn[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
THRB P10828 1/20 0.36
DHODH Q02127 4/20 0.35
CYP2C9 P11712 2/20 0.35
RECQL P46063 1/20 0.34
ABCB11 O95342 1/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADRB3 P13945 1/20 0.34
ADRA2B P18089 1/20 0.34
SLC6A2 P23975 1/20 0.34
TBXAS1 P24557 1/20 0.34
HTR2C P28335 1/20 0.34
AGTR1 P30556 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8417917 0.92 TSHR (0.39) MEN1POLBKMT2ASMN1; SMN2CYP2C9
SCHEMBL8421711 0.91 AGTR1 (0.41) KDM4EKMT2ASMN1; SMN2CYP2C9ABCB11
SCHEMBL8419029 0.90 AGTR1 (0.37) CYP2C9ABCB11EGFRERBB2CYP3A4
SCHEMBL8419094 0.86 MAPT (0.37) KDM4EPOLBSMN1; SMN2DHODHRECQL
SCHEMBL8419225 0.86 DHODH (0.35) POLBDHODHRECQL
SCHEMBL8417426 0.85 TSHR (0.37) MEN1POLBKMT2ACYP2C9ABCB11
SCHEMBL8422155 0.84 DHODH (0.38) KDM4EPOLBDHODHRECQL
SCHEMBL7235119 0.84 DHODH (0.43) KDM4EDHODHCYP2C9ABCB11EGFR
SCHEMBL8417957 0.84 ALOX15 (0.41) KDM4EPOLBSMN1; SMN2CYP2C9ABCB11
SCHEMBL8418031 0.84 ABCB11 (0.34) DHODHCYP2C9ABCB11EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763619-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS OR STROKES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-09 US disclosed
US-5705517-A ANGIOTENSIN II ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-06 US disclosed
US-5703110-A HYPOTENSIVE AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-30 US disclosed