SCHEMBL8635787

SCHEMBL8635787

O=C(CBr)Nc1ccccc1C(=O)c1ccccc1Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 1/20 0.57
GABRD O14764 1/20 0.57
GABRA1 P14867 1/20 0.57
GABRB1 P18505 1/20 0.57
GABRG2 P18507 1/20 0.57
GABRB3 P28472 1/20 0.57
GABRA5 P31644 1/20 0.57
GABRA3 P34903 1/20 0.57
GABRA2 P47869 1/20 0.57
GABRB2 P47870 1/20 0.57
GABRA4 P48169 1/20 0.57
GABRE P78334 1/20 0.57
GABRA6 Q16445 1/20 0.57
GABRG1 Q8N1C3 1/20 0.57
GABRG3 Q99928 1/20 0.57
GABRQ Q9UN88 1/20 0.57
MAPK1 P28482 1/20 0.55
ALDH1A1 P00352 2/20 0.51
CYP1A2 P05177 2/20 0.50
CYP2C19 P33261 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10813064 0.87 GABRP (0.76) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL9380266 0.85 GABRP (0.58) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL8577392 0.84 GABRP (0.77) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL31146466 0.83 KMT2A (0.68) ALDH1A1CYP1A2CYP2C19HPGDMEN1
SCHEMBL5456482 0.83 KMT2A (0.68) ALDH1A1CYP1A2CYP2C19HPGDMEN1
SCHEMBL9573562 0.81 ALDH1A1 (0.48) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL30192167 0.81 GABRP (0.54) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL6907111 0.81 GABRP (0.54) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL9652547 0.81 GABRP (0.54) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL8672570 0.81 ALDH1A1 (0.71) MAPK1ALDH1A1HPGDMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5706829-A BENZODIAZEPINE DERIVATIVE CREIGHTON UNIVERSITY (US) 1998-01-13 US disclosed
US-4014883-A ANTITUMOR AGENTS HOFFMANN-LA ROCHE INC. (US) 1977-03-29 US disclosed