SCHEMBL8635985

SCHEMBL8635985

CCN1CCCC1Oc1ccc(C=Cc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 15/20 0.47
CHRNB4 P30926 14/20 0.47
CHRNA3 P32297 14/20 0.47
CHRNA10 Q9GZZ6 7/20 0.46
CHRNA9 Q9UGM1 7/20 0.46
CHRNB2 P17787 10/20 0.46
CHRNA4 P43681 10/20 0.46
RELA Q04206 1/20 0.45
LTA4H P09960 1/20 0.44
TRPA1 O75762 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
THPO P40225 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7246918 0.87 CARM1 (0.40) CHRNA7CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL4322788 0.83 MEN1 (0.39)
SCHEMBL8641764 0.82 HRH3 (0.50) LTA4H
SCHEMBL7397894 0.82 MAOA (0.47) CHRNA7CHRNB4CHRNA3CHRNA10CHRNA9
Hydrochloric Acid SCHEMBL7402438 0.81 MAOA (0.46) CHRNA7CHRNB4CHRNA3CHRNA10CHRNA9
SCHEMBL8641777 0.80 HRH3 (0.57) CHRNA7CHRNB2CHRNA4LTA4H
SCHEMBL8147094 0.79 ATM (0.44) CHRNA7CHRNB2CHRNA4
SCHEMBL8637445 0.78 HRH1 (0.46) LTA4H
SCHEMBL11277901 0.77 HRH3 (0.42)
SCHEMBL8640957 0.75 LTA4H (0.41) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed