SCHEMBL8637017

SCHEMBL8637017

Cc1ccccc1S(=O)(=O)OC(C)c1ccc(C(C(=O)O)C2CCCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HTR1E P28566 2/20 0.40
S1PR3 Q99500 2/20 0.40
CHRM3 P20309 3/20 0.39
LMNA P02545 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
EPHX2 P34913 1/20 0.39
CYP3A4 P08684 2/20 0.38
CYP1A2 P05177 2/20 0.38
TSHR P16473 2/20 0.38
CHRM2 P08172 1/20 0.38
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38
CHRM1 P11229 1/20 0.38
DRD1 P21728 1/20 0.38
SLC6A2 P23975 1/20 0.38
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637023 0.81 ALOX5 (0.40) ALOX5HDAC6HTR1ES1PR3CHRM3
SCHEMBL8639290 0.79 CHRM3 (0.41) ALOX5HDAC6CHRM3LMNACYP3A4
SCHEMBL69127 0.72 HTR1E (0.65) ALOX5HDAC6HTR1ES1PR3CHRM3
SCHEMBL28622389 0.72 HTR1E (0.65) ALOX5HDAC6HTR1ES1PR3CHRM3
SCHEMBL8960414 0.72 CYP1A2 (0.46) MEN1KMT2ACYP1A2TSHRCYP2C9
SCHEMBL8960400 0.72 CYP1A2 (0.46) MEN1KMT2ACYP1A2TSHRCYP2C9
SCHEMBL1177706 0.71 HTR1E (0.60) ALOX5HDAC6HTR1ES1PR3CHRM3
SCHEMBL1177709 0.71 HTR1E (0.60) ALOX5HDAC6HTR1ES1PR3CHRM3
SCHEMBL12531975 0.71 HTR1E (0.63) ALOX5HTR1ES1PR3CHRM3LMNA
SCHEMBL67219 0.71 HTR1E (0.63) ALOX5HTR1ES1PR3CHRM3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776964-A HYPOTENSIVE AGENTS; ANTICHOLESTEROL AGENTS; CARDIOVASCULAR DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1998-07-07 US disclosed
US-5521206-A HYPOTENSIVE AGENTS, TREATMENT OF ATHEROSCLEROSIS BAYER AKTIENGESELLSCHAFT (DE) 1996-05-28 US disclosed