SCHEMBL8637152

SCHEMBL8637152

COc1ccc(CC(=O)Nc2ccccc2C(N)=O)cc1OC

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.64
POLB P06746 2/20 0.64
GFER P55789 1/20 0.64
KMT2A Q03164 4/20 0.63
LMNA P02545 4/20 0.63
MEN1 O00255 2/20 0.63
SMN1; SMN2 Q16637 2/20 0.62
RAB9A P51151 1/20 0.60
ATM Q13315 1/20 0.60
EPHX2 P34913 1/20 0.59
KDM4E B2RXH2 2/20 0.57
HTT P42858 1/20 0.57
PARP14 Q460N5 1/20 0.57
BCHE P06276 1/20 0.57
ACHE P22303 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8639241 0.93 KDM4E (0.60) GAAPOLBGFERKMT2ALMNA
SCHEMBL28618230 0.91 CHEK1 (0.63) GAAPOLBGFERKMT2ALMNA
SCHEMBL28607272 0.91 GAA (0.70) GAAPOLBGFERKMT2ALMNA
SCHEMBL28607667 0.89 POLB (0.64) GAAPOLBGFERKMT2ALMNA
SCHEMBL8638027 0.88 MEN1 (0.67) GAAPOLBGFERKMT2ALMNA
SCHEMBL1645810 0.88 KMT2A (0.71) GAAPOLBGFERKMT2ALMNA
SCHEMBL8637193 0.87 KMT2A (0.60) GAAKMT2ALMNAMEN1SMN1; SMN2
SCHEMBL8639573 0.83 RAB9A (0.70) GAAPOLBKMT2AMEN1SMN1; SMN2
SCHEMBL8638900 0.83 MAPK8 (0.65) GAAPOLBKMT2ALMNAMEN1
SCHEMBL8639229 0.81 MAPT (0.71) GAAGFERKMT2ALMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855387-A1 2-ACYLAMINOBENZAMIDE DERIVATIVES AND PREVENTIVE AND REMEDY FOR DISEASES CAUSED BY THE SUPERMULTIPLICATION OF VASCULAR INTIMAL CELLS KISSEI PHARMACEUTICAL CO., LTD. (JP) 1998-07-29 EP disclosed