SCHEMBL8638263

SCHEMBL8638263

Clc1cccc(CC2CCN(CCOc3ccccc3)C2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 2/20 0.65
SIGMAR1 Q99720 2/20 0.65
HTT P42858 2/20 0.57
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
GLA P06280 1/20 0.57
GAA P10253 1/20 0.57
MAPT P10636 1/20 0.57
ATM Q13315 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
LMNA P02545 1/20 0.56
MAPK1 P28482 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
LTA4H P09960 6/20 0.53
HTR1A P08908 2/20 0.53
HTR7 P34969 2/20 0.53
HRH3 Q9Y5N1 1/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A4 P31645 1/20 0.52
KMT2A Q03164 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8639262 0.87 SIGMAR1 (0.70) TMEM97SIGMAR1ALDH1A1LTA4HHTR1A
SCHEMBL8637770 0.86 TMEM97 (0.65) TMEM97SIGMAR1LTA4HHTR1AHTR7
SCHEMBL8641102 0.86 HTR1A (0.67) TMEM97SIGMAR1GAALTA4HHTR1A
SCHEMBL7248846 0.80 TMEM97 (0.71) TMEM97SIGMAR1HTTLTA4HHRH3
SCHEMBL5888854 0.80 TMEM97 (1.00) TMEM97SIGMAR1KDM4EALDH1A1SMN1; SMN2
SCHEMBL8644124 0.80 TMEM97 (0.70) TMEM97SIGMAR1LTA4HHTR1AHTR7
Bromide SCHEMBL7253600 0.79 TMEM97 (0.69) TMEM97SIGMAR1HTTLTA4HHRH3
SCHEMBL7406605 0.79 SIGMAR1 (0.82) TMEM97SIGMAR1KDM4EALDH1A1SMN1; SMN2
SCHEMBL7409069 0.79 SIGMAR1 (0.82) TMEM97SIGMAR1KDM4EALDH1A1SMN1; SMN2
SCHEMBL2158157 0.79 KCNH2 (0.63) TMEM97SIGMAR1HTTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed