SCHEMBL8639345

SCHEMBL8639345

NS(=O)(=O)c1ccccc1-n1nc(C(F)F)cc1C1=CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.47
PTGS1 P23219 9/20 0.43
SLC5A1 P13866 1/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 1/20 0.34
PTGES2 Q9H7Z7 1/20 0.34
ABCB11 O95342 1/20 0.34
ALDH1A1 P00352 1/20 0.34
FFAR2 O15552 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8641648 0.83 PTGS2 (0.69) PTGS2PTGS1
SCHEMBL8693450 0.82 PTGS2 (0.44) PTGS2PTGS1CA12CA1CA2
SCHEMBL6013908 0.81 PTGS2 (0.71) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8641235 0.80 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8692227 0.80 PTGS2 (0.44) PTGS2PTGS1CA12CA1CA2
SCHEMBL7928751 0.79 PTGS2 (0.66) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8637047 0.78 PTGS2 (0.63) PTGS2PTGS1CA1CA2CA9
SCHEMBL7773921 0.76 PTGS2 (0.65) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8525009 0.76 PTGS2 (0.65) PTGS2PTGS1CA12CA1CA2
SCHEMBL8637387 0.75 PTGS2 (0.54) PTGS2PTGS1ABCB11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed