SCHEMBL8639693

SCHEMBL8639693

CC(=O)c1cc(C(=O)O)ccc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.50
LMNA P02545 2/20 0.50
MAPK1 P28482 1/20 0.50
HTT P42858 1/20 0.50
KDM4E B2RXH2 4/20 0.47
TSHR P16473 3/20 0.47
GAA P10253 2/20 0.47
ALDH1A1 P00352 1/20 0.47
AKR1C3 P42330 5/20 0.44
AKR1C2 P52895 5/20 0.44
AKR1B10 O60218 1/20 0.43
AKR1B1 P15121 1/20 0.43
AKR1C4 P17516 1/20 0.43
AKR1C1 Q04828 1/20 0.43
TP53 P04637 1/20 0.42
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA4 P22748 2/20 0.42
CA6 P23280 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL336060 0.85 KDM4E (0.52) RAB9ALMNAMAPK1HTTKDM4E
SCHEMBL17478757 0.84 AKR1C3 (0.53) AKR1C3AKR1C2AKR1B10AKR1B1AKR1C4
SCHEMBL19331714 0.84 RAB9A (0.55) RAB9ALMNAMAPK1HTTKDM4E
SCHEMBL10316500 0.82 PARP1 (0.46) KDM4EALDH1A1CA1CA2CES2
SCHEMBL7898447 0.81 KDM4E (0.52) RAB9AKDM4ETSHRGAAALDH1A1
SCHEMBL27952405 0.80 LMNA (0.46) RAB9ALMNAMAPK1HTTKDM4E
SCHEMBL23263412 0.79 GAA (0.55) RAB9ALMNAMAPK1HTTKDM4E
SCHEMBL1815890 0.79 RAB9A (0.54) RAB9ALMNAMAPK1HTTKDM4E
SCHEMBL8641593 0.79 ALDH1A1 (0.54) RAB9ALMNAHTTKDM4EGAA
SCHEMBL1602112 0.79 RAB9A (0.46) RAB9ALMNAMAPK1HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102153535-A Benzopyranyl-3-alcohol esterified derivative serving as antineoplastic multidrug resistance inhibitor and preparation method and application of benzopyranyl-3-alcohol esterified derivative OCEAN UNIV CHINA 2011-08-17 CN disclosed
US-5849775-A Substituted benzoylguanidines process for their preparation, their use as a medicament or diagnostic, and pharmaceutical containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-12-15 US disclosed
US-5679712-A ANTIARRHYTHMIA AGENTS, TREATMENT OF CARDIOVASCULAR, NERVOUS SYSTEM DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-10-21 US disclosed
US-5631293-A CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-20 US disclosed