SCHEMBL8640401

SCHEMBL8640401

CS(=O)(=O)c1ccc(-n2nc(C(F)(F)Cl)cc2-c2ccc(F)cc2)cc1

nearest known ligand 0.82

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.82
PTGS1 P23219 6/20 0.82
CYP2C9 P11712 1/20 0.67
AOC3 Q16853 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9003005 0.90 PTGS2 (0.67) PTGS2PTGS1CYP2C9
SCHEMBL5229949 0.90 PTGS2 (1.00) PTGS2PTGS1CYP2C9
Sc-58125 SCHEMBL214120 0.90 PTGS2 (1.00) PTGS2PTGS1CYP2C9
Sc-58125 SCHEMBL12375146 0.90 PTGS2 (1.00) PTGS2PTGS1CYP2C9
SCHEMBL9002935 0.89 PTGS2 (0.82) PTGS2PTGS1CYP2C9
SCHEMBL9003167 0.89 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL9260744 0.89 PTGS2 (0.81) PTGS2PTGS1CYP2C9
SCHEMBL9003046 0.88 PTGS2 (0.82) PTGS2PTGS1CYP2C9AOC3
SCHEMBL9002595 0.86 PTGS2 (0.78) PTGS2PTGS1CYP2C9AOC3
SCHEMBL8953925 0.86 PTGS2 (0.78) PTGS2PTGS1CYP2C9AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731793-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP claimed
WO-1995015315-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO claimed
EP-0830133-A1 THERAPEUTIC COMPOSITION FOR ARTHRITIS Takeda Chemical Industries, Ltd. (JP) 1998-03-25 EP disclosed
WO-1996033717-A1 THERAPEUTIC COMPOSITION FOR ARTHRITIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-31 WO disclosed
EP-0731793-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP disclosed
US-5475018-A Antiinflammatory agent, antiarthritic agent; analgesics and antipyretics G. D. SEARLE & CO. (US) 1995-12-12 US disclosed
WO-1995015315-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO disclosed