SCHEMBL9003167

SCHEMBL9003167

CS(=O)(=O)c1ccc(-n2nc(C(F)(F)Cl)cc2-c2ccc(Br)cc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.65
PTGS1 P23219 3/20 0.65
CYP2C9 P11712 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8953883 0.90 PTGS2 (0.80) PTGS2PTGS1CYP2C9
SCHEMBL6516184 0.90 PTGS2 (0.80) PTGS2PTGS1CYP2C9
SCHEMBL9003005 0.89 PTGS2 (0.67) PTGS2PTGS1CYP2C9
SCHEMBL8640401 0.89 PTGS2 (0.82) PTGS2PTGS1CYP2C9
SCHEMBL9002935 0.88 PTGS2 (0.82) PTGS2PTGS1CYP2C9
SCHEMBL9003244 0.88 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL9260744 0.88 PTGS2 (0.81) PTGS2PTGS1CYP2C9
SCHEMBL9256036 0.86 PTGS2 (0.63) PTGS2PTGS1CYP2C9
SCHEMBL8420730 0.81 PTGS2 (0.88) PTGS2PTGS1CYP2C9
SCHEMBL8953923 0.81 PTGS2 (0.80) PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731793-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP claimed
WO-1995015315-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO claimed
US-5475018-A Antiinflammatory agent, antiarthritic agent; analgesics and antipyretics G. D. SEARLE & CO. (US) 1995-12-12 US disclosed