SCHEMBL9002935

SCHEMBL9002935

CS(=O)(=O)c1ccc(-n2nc(C(F)(F)Cl)cc2-c2ccc(I)cc2)cc1

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.82
PTGS1 P23219 3/20 0.65
CYP2C9 P11712 2/20 0.65
PDPK1 O15530 3/20 0.52
ALOX5 P09917 2/20 0.52
PTGES O14684 1/20 0.52
HDAC3 O15379 1/20 0.52
CA12 O43570 1/20 0.52
PDE5A O76074 1/20 0.52
ABCB11 O95342 1/20 0.52
MT-CO2 P00403 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
LMNA P02545 1/20 0.52
CA3 P07451 1/20 0.52
CYP3A4 P08684 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
CYP2D6 P10635 1/20 0.52
ADRB3 P13945 1/20 0.52
ALOX15 P16050 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8953873 0.90 PTGS2 (1.00) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL8636647 0.90 PTGS2 (1.00) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL9003005 0.89 PTGS2 (0.67) PTGS2PTGS1CYP2C9PDPK1CYP3A4
SCHEMBL8640401 0.89 PTGS2 (0.82) PTGS2PTGS1CYP2C9
SCHEMBL9003167 0.88 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL8635653 0.88 PTGS2 (0.82) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL9260744 0.88 PTGS2 (0.81) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL9002988 0.86 PTGS2 (0.79) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL8635490 0.81 PTGS2 (0.80) PTGS2PTGS1CYP2C9PDPK1CYP3A4
SCHEMBL8953923 0.81 PTGS2 (0.80) PTGS2PTGS1CYP2C9PDPK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731793-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP claimed
WO-1995015315-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO claimed
US-5475018-A Antiinflammatory agent, antiarthritic agent; analgesics and antipyretics G. D. SEARLE & CO. (US) 1995-12-12 US disclosed