SCHEMBL8640755

SCHEMBL8640755

Fc1ccc([C]2CCNC2)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.40
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
TDP2 O95551 1/20 0.36
PARP10 Q53GL7 1/20 0.36
GRM5 P41594 1/20 0.35
ACKR3 P25106 1/20 0.35
ALDH1A1 P00352 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
PIK3CG P48736 1/20 0.34
MELK Q14680 1/20 0.33
HTR6 P50406 1/20 0.33
NISCH Q9Y2I1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL434353 0.79 ALDH1A1 (0.42) TDP2ALDH1A1PDE3BPDE3A
SCHEMBL16518134 0.78 PARP1 (0.41) PARP1HTR2AHTR2CPDE3BPDE3A
SCHEMBL8355517 0.76 HTR7 (0.46) HTR2CALDH1A1HTR6NISCH
SCHEMBL436723 0.75 MAOA (0.41) TDP2ALDH1A1
SCHEMBL435076 0.75 ALDH1A1 (0.39) TDP2ALDH1A1
SCHEMBL16518151 0.74 PNMT (0.46) PARP1HTR2AHTR2CHTR6NISCH
SCHEMBL16518127 0.74 PRCP (0.55) PARP1
SCHEMBL16518161 0.74 PARP1 (0.39) PARP1HTR2AHTR2CPDE3BPDE3A
SCHEMBL16492225 0.74 PKN2 (0.51) PARP1HTR2AHTR2CTDP2PARP10
SCHEMBL8635851 0.74 HTR2A (0.42) HTR2AHTR2CHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed