SCHEMBL8640822

SCHEMBL8640822

CS(=O)(=O)c1ccc(-c2[nH]nc(Cl)c2-c2ccc(C#N)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.49
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
PTGS1 P23219 2/20 0.40
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637748 0.85 PTGS2 (0.56) PTGS2PTGS1
SCHEMBL8067283 0.82 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL8074136 0.79 EPAS1 (0.42) PTGS2PTGS1
SCHEMBL8069284 0.77 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL3865448 0.76 PTGS2 (0.40) PTGS2CYP11B1CYP11B2CA12CA1
SCHEMBL4190362 0.75 PTGS2 (0.72) PTGS2CYP11B1CYP11B2CA12CA1
SCHEMBL8068397 0.75 PTGS2 (0.53) PTGS2
SCHEMBL8058037 0.74 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL803901 0.73 PTGS2 (0.68) PTGS2CYP11B1CYP11B2CA12CA1
Isophthalic Acid SCHEMBL27322237 0.73 CSNK2A1 (0.41) PTGS2CYP11B1CYP11B2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0856000-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-08-05 EP disclosed
WO-1997013755-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-04-17 WO disclosed