SCHEMBL8644469

SCHEMBL8644469

O=C1CN(CCC(c2ccccc2)N2CCOCC2)S(=O)(=O)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.50
KMT2A Q03164 3/20 0.44
CTDSP1 Q9GZU7 2/20 0.44
MDM2 Q00987 1/20 0.44
TSHR P16473 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ACHE P22303 1/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 2/20 0.37
PIK3CD O00329 1/20 0.37
PIK3R2 O00459 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
PIK3R5 Q8WYR1 1/20 0.37
PIK3R3 Q92569 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KCNA5 P22460 1/20 0.36
ATM Q13315 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8648976 0.99 TDP1 (0.49) TDP1KMT2ACTDSP1MDM2TSHR
SCHEMBL8644541 0.80 ACHE (0.46) TDP1KMT2ACTDSP1MDM2TSHR
Hydrochloric Acid SCHEMBL8646984 0.80 ACHE (0.46) TDP1KMT2ACTDSP1MDM2TSHR
SCHEMBL8646533 0.77 TDP1 (0.53) TDP1KMT2ACTDSP1MDM2TSHR
SCHEMBL8645313 0.74 TDP1 (0.50) TDP1KMT2ACTDSP1MDM2TSHR
Fumaric Acid SCHEMBL8649180 0.73 TDP1 (0.49) TDP1KMT2ACTDSP1MDM2TSHR
Fumaric Acid SCHEMBL8649177 0.73 TDP1 (0.49) TDP1KMT2ACTDSP1MDM2TSHR
SCHEMBL8645472 0.73 DRD2 (0.42) TDP1KMT2ATSHRSMN1; SMN2ACHE
Ethylene SCHEMBL8646719 0.72 TDP1 (0.48) TDP1KMT2ACTDSP1MDM2TSHR
SCHEMBL8648315 0.72 DRD2 (0.56) TDP1KMT2ACTDSP1MDM2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773437-A UROGENITAL DISORDERS SUCH AS DYSURIA NIPPON CHEMIPHAR CO., LTD. (JP) 1998-06-30 US disclosed
EP-0753514-A1 ALKYLENEDIAMINE DERIVATIVE NIPPON CHEMIPHAR CO., LTD. (JP) 1997-01-15 EP disclosed