SCHEMBL8647153

SCHEMBL8647153

COc1ccccc1/C=C(/C(=O)NC(=N)NOS(C)(=O)=O)c1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 3/20 0.47
CYP1A2 P05177 3/20 0.47
CYP1B1 Q16678 3/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
CAPN1 P07384 1/20 0.46
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
POLB P06746 2/20 0.42
MAPT P10636 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 4/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 2/20 0.37
ATM Q13315 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8650931 0.89 ATM (0.37) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL8646248 0.88 MAPT (0.43) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL8648668 0.88 ALDH1A1 (0.35) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL8647149 0.87 CYP1A1 (0.50) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL8650932 0.85 NPC1 (0.42) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL8644572 0.85 CYP1A1 (0.54) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL8648674 0.84 KMT2A (0.47) CYP3A4POLBMAPTNPC1RAB9A
SCHEMBL8644322 0.81 MAPT (0.42) CYP3A4MAPTNPC1RAB9AKMT2A
SCHEMBL8646761 0.80 CYP3A4 (0.45) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL8646382 0.77 CYP1A1 (0.46) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861831-A1 HETEROARYL-SUBSTITUTED ACRYLOYLGUANIDINE DERIVATIVES AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-09-02 EP disclosed